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SB 218795
CAS No. 174635-53-1
SB 218795 ( —— )
产品货号. M27703 CAS No. 174635-53-1
SB 218795 is an effective and selective antagonist of NK3 with a Ki 13 nM for hNK3 which is about 90-fold and 7000-fold selectivity over hNK2 and hNK1.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥786 | 有现货 |
|
| 10MG | ￥1393 | 有现货 |
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| 25MG | ￥2811 | 有现货 |
|
| 50MG | ￥4560 | 有现货 |
|
| 100MG | ￥6423 | 有现货 |
|
| 500MG | ￥13527 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称SB 218795
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述SB 218795 is an effective and selective antagonist of NK3 with a Ki 13 nM for hNK3 which is about 90-fold and 7000-fold selectivity over hNK2 and hNK1.
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产品描述SB 218795 is an effective and selective antagonist of NK3 with a Ki 13 nM for hNK3 which is about 90-fold and 7000-fold selectivity over hNK2 and hNK1.(In Vitro):SB 218795 (3-30 nM) antagonizes the contractile responses senktide-induced in a surmountable and concentration-dependent manner.(In Vivo):In rabbits, SB?218795 (0.25-1?mg/kg; i.v.) inhibits NK3 receptor-mediated pupillary constriction by maximum inhibition of 78%.
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同义词——
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通路GPCR/G Protein
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靶点Neurokinin Receptor
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受体——
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研究领域——
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适应症——
化学信息
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CAS Number174635-53-1
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分子量396.4
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分子式C25H20N2O3
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纯度>98% (HPLC)
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溶解度——
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SMILESCOC(=O)[C@@H](NC(=O)c1cc(nc2ccccc12)-c1ccccc1)c1ccccc1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Carnat A1, et al. Luteolin 7-diglucuronide, the major flavonoid compound from Aloysia triphylla and Verbena officinalis.Planta Med. 1995 Oct;61(5):490.
产品手册
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